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Drug Intermediates

VARDA Biotech, delivers its Strategic outsourcing services through the Pharmaceutical Division, which is having domestic and international horizontals, as separate entities.

We deliver our services for Global Markets in Exporting Active Pharmaceutical Ingredients and Drug Intermediates through our Global Pharmaceuticals Business Unit.

For any requirement of the Pharmaceutical Bulk Drugs/Drug Intermediates, please contact Contact Us

 

DRUG INTERMEDIATE LIST

SEGMENTED Chemistry GROUP /

DRUG ACTIVE (API)

DRUG INTERMEDIATES

 
AZOLE CHEMISTRY
PRODUCTS CAS NO APPLICATION

5-Methoxy-2-(4-methoxy-3,5-dimethylpyridine-2yl)methylthio)-1H-benzimidazole

73590-85-9

Es-Omeprazole / Omeprazole

 

2-Chloro methyl-3-methyl-4 (2,2,2-tri flouro ethoxy) pyridine hydrochloride

127337-60-4

Lansoprazole

 

2-Chloromethyl-4-Methoxy-3,5-Dimethyl Pyridine HCl

86604-75-3

Omeprazole

 

5-Difluro Methoxy-2-[[(3,4-Dimethoxy-2-Pyridinyl)Methyl]Thio]-1H-Benzimidazole (Sulphide)

102625-64-9

Pantoprazole

 

3-Methoxy-1-Propanol

1589-49-7

Rabeprazole

2-(Chloromethyl)-4-(3-Methoxy Propoxy)-3-Methyl Pyridine HCl

153259-31-5

Rabeprazole

 

2-({[4-(3-Methoxy Propoxy)-3-Methyl Pyridine-2-YL] Methyl} Sulfa)1H-Benzimidazole 2,3-Dimethyl-4-Nitro Pyridine-N-Oxide

117977-21-6

Rabeprazole

 

4-Chloro-6-ethyl-5-fluoro pyrimidine

 

Voriconazole Posoconazole

1-(2,3) Dichlorophenyl) Piperazine Base

119532-26-2

Aripiprazole

7-Hydroxy-3,4-Carbostyril

 

Aripiprazole

ANTIRETROVIRAL CHEMISTRY
PRODUCTS CAS NO APPLICATION

2,5-Diamino-4,6-Dihydroxy Pyrimidine Hydrochloride Monohydrate (DAPDIOL)

 

Abacavir

N-(2-Amino-4,6-Dichloropyrimidine-5-yl)Formamide (FADCP)

 

Abacavir

4,6-Dichloropyrimidine-2,5-Diamine (DADCP)

 

Abacavir

(S)-5-Chloro-alpha-(Cyclopropylethynyl)-2-amino-alpha-(trifluoromethyl) benzene methanol   Efavirenz

(S)-5-chloro-a-(cyclopropylethenyl)-2-[((4-methoxyphenyl)methyl)amino]- a-(trifluoromethyl)benzene methanol

 

Efavirenz

2-Isopropyl-5R-Methyl Cyclohexyl-2-Oxo-Acetate

 

Lamivudine

2-(2S-Isopropyl-5R-Methyl-1R-Cyclohexyl)-5-Hydroxy-1,3-Oxathilan-2-Carboxalate

 

Lamivudine

2-5-Isopropyl-5R-Methyl-1R-Cyclohexyl ester-(1,3)-Oxathiolan-5-Hydroxy-2-Carboxate

 

Lamivudine

(2R-Cis)-4-Amino-1-[2-(hydroxy methyl)-1,3-Oxathilolan-5-yl]-2-(1H) Pyrimidinone

 

Lamivudine

2-Chloro-N-[2-chloro-4-methyl pyridinyl]-3- pyridine carboxamide

 

Nevirapine

5-Benzoyl-2,3-Didehydro-3-deoxythymidine

 

Stauvidine

Stauvidine NMPO Solvate

 

Stauvidine

N-1-(Tertiarybutyl oxy carbonyl)N-2-[4-(Pyridine-2-yl)Benzylidene]-Hydrazine

 

Atazenavir

N-1-(Tertiarybutyl oxy carbonyl)-2 (S)-Amino-1-Phenyl-3(R)-3,4-Epoxy Butane (Under Development)

 

Atazenavir

 
 
   

CNS Chemistry

PRODUCTS CAS NO APPLICATION

3-Dimethyl amino-1- (2-thienyl)-1-propanone hydrochloride

 

Duloxetine

RS-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)-1-propanamine

116817-84-6

Duloxetine

S(+)-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)-1-propanamine

 

Duloxetine

RS-N,N- Dimethyl-3-(1-Naphthalenyloxy)-3-(2-thienyl)-1-propanamine oxalate

 

Duloxetine

S(+)-N,N- Dimethyl-3-(1-Naphthalenyloxy)-3-(2-thienyl)-1-propanamine oxalate

132335-47-8

Duloxetine

5,6-Dimethoxy Indanone

2107-69-9

Donepezil

1-Benzyl-4-Piperidine Carboxyaldehyde

22065-85-6

Donepezil

1-Benzyl-4-Piperidine Methanol HCl

67686-01-5

Donepezil

5-Nitro Vanilline

6635-20-7

Entacapone

3,4-Dihydroxy-5-nitro benzaldehyde

116313-85-0

Entacapone

N,N-Diethyl-2-Cyano Acetamide

26391-06-0

Entacapone

2,3-Dichloro Benzoyl Nitrile

77668-42-9

Lamotrigene

Diphenyl Methyl Thio Acetamide

68524-30-1

Modafinil

(±) Diphenyl Methane Sulfinyl Acetic Acid

 

Modafinil

(±) [2-(Diphenyl) Methane Sulfinyl] Acetamide

 

Modafinil

(±)-3-(Aminomethyl)-5-methylhexanoic acid

 

Pregabalin

1,2,2-hydroxy ethoxy ethyl piperazine

13349-82-1

Quetiapine Hemifumarate

Dibenzo-[b,f][1,4] Thiazepin-11-yl] piperazine Dihydrochloride

3159-07-7

Quetiapine Hemifumarate

2-Bromoethyl Benzaldehyde

 

Ropinirole

4-(2-Bromoethyl)-3-Chloro-1,3-Dihydro-2H-Indole-2-One

 

Ropinirole

4-(2-Bromoethyl)-1,3-Dihydro-2H-Indole-2-One

 

Ropinirole

Ethyl methyl carbamic acid-3-((S)-1-dimethylamino ethyl)phenyl ester   Rivastigmine

N-ethyl-N-methyl-carbomyl chloride (RV-I)

 

Rivastigmine

3-(1-Diethylaminoethyl)Phenol HCl (RV-II)

105601-04-5

Rivastigmine

(S)-1(3-hydroxyphenyl)-N,N-dimethyl ethyl amine

 

Rivastigmine

Tetralone (4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-naphthalenone)

79560-19-3

Sertraline HCl

1,2-Benzisoxazole-3-Methane Sulfonic Acid Sodium Salt

73101-64-1

Zonisamide

2-amino-5-chloro pyridine

1072-98-6

Zopiclone

6-(5-chloropyrid-2-yl)-5-hydroxy-7-oxo-5,6-dihydro pyrrolo[3,4-b]-pyrazine

 

Zopiclone

6-(5-chloropyrid-2-yl)-5,7-dioxo-5,6-dihydropyrrolo-[3,4-b]-pyrazine

 

Zopiclone

   
ONCOLOGY CHEMISTRY
PRODUCTS CAS NO APPLICATION

4-Amino-2-Trifluoromethyl Benzonitrile

654-70-6

Bicalutamide

4-Cyano-N-Methacryloyl-3-Trifluoro Methyl Aniline

90357-53-2

Bicalutamide

N-[4-Cyano-3-(Trifluoromethyl)Phenyl]-3-[(4-Fluorophenyl)Thio]-2-Hydroxy-2-Methyl Propanamide- (Sulphide)

90356-78-8

Bicalutamide

6,7-Dimethoxy Quinozoline-4-one

 

Geftinib

(D-erythro)-2-Deoxy-2,2-Difluoro pentafuranose-1-ulose-3,5- dibenzoate                    

122111-01-7

Gemcitabine

2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate

143157-22-6

Gemcitabine

2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-di benzoate-1-methane sulfonate

122111-11-9

Gemcitabine

10-Hydroxy –7 – Ethyl Comptothecin

64439-81-2

Irinotecan

4-Piperidino Piperidine

4897-50-1  

Irinotecan

4-Piperdino Piperdine Corbomile Chloride HCl

 

Irinotecan

N-Methyl Pentylamine

 

Ibandronate

4[(4-Methyl Piperazino)Methyl Benzoic Acid

 

Imatinib Mesylate

3-Pyridyl Acetic Acid Hydrochloride

6419-36-9

Risedronate Sodium

   
PRIL CHEMISTRY
PRODUCTS CAS NO APPLICATION

 g - Benzyl Glutamate

  Cilazaril

[2- methyl -1-(1- oxo propoxy) propoxy](4- phenyl butyl) phosphinyl] acetic acid.    

123599-78-0

Fosinopril

Trans-4-cyclohexyl-L-Proline

103201-78-1

Fosinopril

Hydroxy-(4-Phenylbutyl)-phosphonic acetic acid phenyl methyl ester

 

Fosinopril

Diasteromeric mixture of Octahydro-1H-indole-2-carboxylic acid [( 3aR, 7aS)/ (2R, 3aS, 7aR)]

 

Perindopril

(2S,3aS,7aS)Octahydroindole-2-carboxylic acid benzyl ester hydrochloride

 

Perindopril

TIQ-Benz-pTSA salt (QL-2) (PhenylMethyl(3S)-1,2,3,4-Tetrahydroisoquinoline-3-Carboxylate.pTSA)

 

Quinapril

Quinapril Benzyl Ester

 

Quinapril

Chloro Serene N-Acetyl Methyl Ester

 

Ramipril

Benzyl Cis Endo Octa Hydro Penta Pyrrole-2-Carboxylate HCl

 

Ramipril

Carboethoxy-3-Phenl Propylalanine Cis Endo Octahydro Cyclopenta (b) Pyrrole Benzyl Carboxylate

 

Ramipril

   

SARTAN CHEMISTRY

PRODUCTS CAS NO APPLICATION
Methyl-2-(tert-butoxy carbonyl amino)-3-nitro benzoate   Candesartan

Methyl-2-(tert-butoxy carbonyl amino)-3-nitro benzoate

 

Candesartan